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Compounds

COMPOUND NPA029289

STRUCTURE
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PROPERTIES
NPAID NPA029289
CLUSTER ID 6377
NODE ID 141
NAME Leucinostatin NPDG C
FORMULA C61H111N11O12
MOLECULAR WEIGHT (Da) 1190.6240
ACCURATE MASS (Da) 1189.8414
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Ophiocordyceps
ORIGIN SPECIES sp. and Purpureocillium sp.
InChIKey UTOJVRFQBVCQEH-ZAPMAATISA-N
InChI InChI=1S/C61H111N11O12/c1-20-22-23-42(73)30-39(10)31-45(66-54(80)46-32-40(11)34-72(46)48(75)25-24-38(9)21-2)52(78)68-49(50(76)37(7)8)55(81)70-60(15,16)57(83)67-43(28-35(3)4)51(77)65-44(29-36(5)6)53(79)69-61(17,18)58(84)71-59(13,14)56(82)63-27-26-47(74)64-41(12)33-62-19/h24-25,35-46,49-50,62,73,76H,20-23,26-34H2,1-19H3,(H,63,82)(H,64,74)(H,65,77)(H,66,80)(H,67,83)(H,68,78)(H,69,79)(H,70,81)(H,71,84)/b25-24+/t38-,39+,40-,41-,42+,43-,44-,45-,46-,49-,50+/m0/s1
SMILES CCCC[C@@H](O)C[C@@H](C)C[C@H](NC(=O)[C@@H]1C[C@H](C)CN1C(=O)/C=C/[C@@H](C)CC)C(=O)N[C@H](C(=O)NC(C)(C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NC(C)(C)C(=O)NC(C)(C)C(=O)NCCC(=O)N[C@@H](C)CNC)[C@H](O)C(C)C
ORIGINAL ISOLATION REFERENCE
CITATION Cichewicz, Robert H.; Kil, Yun-Seo; Mooberry, Susan L.; Petersen, Cora L.; Risinger, April L. Leucinostatins from Ophiocordyceps spp. And Purpureocillium spp. Demonstrate Selective Antiproliferative Effects in Cells Representing the Luminal Androgen Receptor Subtype of Triple Negative Breast Cancer Journal of Natural Products 2020 83 (6) 2010-2024.
DOI 10.1021/acs.jnatprod.0c00404 PMID 32510949
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Sordariomycetes MycoBank 147550
Order Hypocreales MycoBank 5125
Family Ophiocordycipitaceae MycoBank 474942
Genus Ophiocordyceps MycoBank 474995
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