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Compounds

COMPOUND NPA024810

STRUCTURE
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PROJECT MOLECULE TO GLOBAL VIEW See Global
EXTERNAL LINKS
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PROPERTIES
NPAID NPA024810
CLUSTER ID None
NODE ID None
NAME Burkholdac B
FORMULA C23H37N3O6S3
MOLECULAR WEIGHT (Da) 547.7650
ACCURATE MASS (Da) 547.1844
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Burkholderia
ORIGIN SPECIES thailandensis
InChIKey VJXBYUITQBTTQM-XMJNTTDOSA-N
InChI InChI=1S/C23H37N3O6S3/c1-4-14(2)21-18(27)12-20(29)32-15-7-5-6-9-34-35-13-17(23(31)26-21)25-22(30)16(8-10-33-3)24-19(28)11-15/h5,7,14-18,21,27H,4,6,8-13H2,1-3H3,(H,24,28)(H,25,30)(H,26,31)/t14-,15+,16-,17-,18+,21-/m1/s1
SMILES CC[C@@H](C)[C@H]1NC(=O)[C@H]2CSSCCC=C[C@@H](CC(=O)N[C@H](CCSC)C(=O)N2)OC(=O)C[C@@H]1O
ORIGINAL ISOLATION REFERENCE
CITATION Biggins JB; Gleber CD; Brady SF Acyldepsipeptide HDAC inhibitor production induced in Burkholderia thailandensis. Organic Letters 2011 13 (6) 1536-1539.
DOI 10.1021/ol200225v PMID 21348454
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Proteobacteria LPSN 1224
Class Betaproteobacteria LPSN 28216
Order Burkholderiales LPSN 80840
Family Burkholderiaceae LPSN 119060
Genus Burkholderia LPSN 32008
REVISIONS
VERSION SMILES CITATION
Original Isolation CCC(C)C1C(CC(=O)OC\2CC(=O)NC(C(=O)NC(CSSCC/C=C2)C(=O)N1)CCSC)O Biggins JB; Gleber CD; Brady SF Acyldepsipeptide HDAC inhibitor production induced in Burkholderia thailandensis. Organic Letters 2011 13 (6) 1536-1539. DOI: 10.1021/ol200225v PMID: 21348454
2 CC[C@@H](C)[C@H]1NC(=O)[C@H]2CSSCCC=C[C@@H](CC(=O)N[C@H](CCSC)C(=O)N2)OC(=O)C[C@@H]1O Benelkebir, Hanae; Donlevy, Alison M; Packham, Graham; Ganesan, A Total synthesis and stereochemical assignment of burkholdac B, a depsipeptide HDAC inhibitor. Organic Letters 2011 13 (24) 6334-7. DOI: 10.1021/ol202197q PMID: 22091906
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