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Compounds

COMPOUND NPA021433

STRUCTURE
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PROPERTIES
NPAID NPA021433
CLUSTER ID 903
NODE ID 782
NAME Papulacandin D
FORMULA C31H42O10
MOLECULAR WEIGHT (Da) 574.6670
ACCURATE MASS (Da) 574.2778
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Papularia
ORIGIN SPECIES sphaerosperma
InChIKey XKSZJTQIZHUMGA-HJHUFFDJSA-N
InChI InChI=1S/C31H42O10/c1-4-19(2)11-7-5-8-12-20(3)23(34)13-9-6-10-14-26(36)40-29-28(37)25(17-32)41-31(30(29)38)27-21(18-39-31)15-22(33)16-24(27)35/h5-6,8-10,12,14-16,19,23,25,28-30,32-35,37-38H,4,7,11,13,17-18H2,1-3H3/b8-5+,9-6+,14-10+,20-12-/t19-,23+,25+,28+,29-,30+,31-/m0/s1
SMILES CC[C@H](C)CC/C=C/C=C(/C)[C@H](O)C/C=C/C=C/C(=O)O[C@H]1[C@H](O)[C@@H](CO)O[C@]2(OCC3=C2C(O)=CC(O)=C3)[C@@H]1O
ORIGINAL ISOLATION REFERENCE
CITATION Traxler P; Gruner J; Auden JA Papulacandins, a new family of antibiotics with antifungal activity, I. Fermentation, isolation, chemical and biological characterization of papulacandins A, B, C, D and E. Journal of Antibiotics 1977 30 (4) 289-296.
DOI 10.7164/antibiotics.30.289 PMID 324958
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Sordariomycetes MycoBank 147550
Order Xylariales MycoBank 37989
Family Apiosporaceae MycoBank 106263
Genus Papularia MycoBank -
SYNTHESES
CITATION 1 Denmark SE; Regens CS; Kobayashi T Total synthesis of papulacandin D. Journal of the American Chemical Society 2007 129 (10) 2774-6. DOI: 10.1021/ja070071z PMID: 17305346
CITATION 2 Denmark SE; Kobayashi T; Regens CS Total Synthesis of (+)-Papulacandin D. Tetrahedron 2010 66 (26) 4745-4759. DOI: 10.1016/j.tet.2010.03.093 PMID: 20711516
REVISIONS
VERSION SMILES CITATION
Original Isolation CC[C@H](C)CC/C=C\C=C(\C)/[C@@H](C/C=C/C=C/C(=O)O[C@H]1[C@@H]([C@H](O[C@]2([C@H]1O)C3=C(C=C(C=C3CO2)O)O)CO)O)O Traxler P; Gruner J; Auden JA Papulacandins, a new family of antibiotics with antifungal activity, I. Fermentation, isolation, chemical and biological characterization of papulacandins A, B, C, D and E. Journal of Antibiotics 1977 30 (4) 289-296. DOI: 10.7164/antibiotics.30.289 PMID: 324958
2 CC[C@H](C)CC/C=C/C=C(/C)[C@H](O)C/C=C/C=C/C(=O)O[C@H]1[C@H](O)[C@@H](CO)O[C@]2(OCC3=C2C(O)=CC(O)=C3)[C@@H]1O Barrett, Anthony G. M.; Peña, Michael; Willardsen, J. Adam Total Synthesis and Structural Elucidation of the Antifungal Agent Papulacandin D. Journal of Organic Chemistry 1996 61 (3) 1082-1100. DOI: 10.1021/jo951895e
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