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Compounds

COMPOUND NPA020953

STRUCTURE
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PROPERTIES
NPAID NPA020953
CLUSTER ID 6575
NODE ID 4555
NAME Vanoxonin
FORMULA C18H25N3O9
MOLECULAR WEIGHT (Da) 427.4100
ACCURATE MASS (Da) 427.1591
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Saccharopolyspora
ORIGIN SPECIES hirsuta MG245-CF2
InChIKey KCWDMHXDGAWLOA-LQJRIPTKSA-N
InChI InChI=1S/C18H25N3O9/c1-9(22)14(20-16(26)11-5-3-7-13(24)15(11)25)17(27)19-12(18(28)29)6-4-8-21(30)10(2)23/h3,5,7,9,12,14,22,24-25,30H,4,6,8H2,1-2H3,(H,19,27)(H,20,26)(H,28,29)/t9-,12+,14+/m1/s1
SMILES C[C@H]([C@@H](C(=O)N[C@@H](CCCN(C(=O)C)O)C(=O)O)NC(=O)C1=C(C(=CC=C1)O)O)O
ORIGINAL ISOLATION REFERENCE
CITATION Kanai F; Sawa T; Hamada M; Naganawa H; Takeuchi T; Umezawa H VANOXONIN, A NEW INHIBITOR OF THYMIDYLATE SYNTHETASE Journal of Antibiotics 1983 36 (6) 656-660.
DOI 10.7164/antibiotics.36.656 PMID 6874588
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Actinobacteria LPSN 201174
Class Actinobacteria LPSN -
Order Pseudonocardiales LPSN 85010
Family Pseudonocardiaceae LPSN 2070
Genus Saccharopolyspora LPSN 1835
SYNTHESES
CITATION 1 Kanai F; Isshiki K; Umezawa Y; Morishima H; Naganawa H; Takita T; Takeuchi T; Umezawa H Vanoxonin, a new inhibitor of thymidylate synthetase. II. Structure determination and total synthesis. Journal of Antibiotics 1985 38 (1) 31-8. DOI: 10.7164/antibiotics.38.31 PMID: 3972726
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