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Compounds

COMPOUND NPA018815

STRUCTURE
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PROPERTIES
NPAID NPA018815
CLUSTER ID 1983
NODE ID 1017
NAME Nominine
FORMULA C28H39NO
MOLECULAR WEIGHT (Da) 405.6260
ACCURATE MASS (Da) 405.3032
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Aspergillus
ORIGIN SPECIES nomius (NRRL 13137)
InChIKey BSSPRCKKWJRAJZ-HBDSXALQSA-N
InChI InChI=1S/C28H39NO/c1-19(2)9-8-15-28-24(17-22-18-29-25-11-7-6-10-23(22)25)20(3)14-16-27(28,5)21(4)12-13-26(28)30/h6-7,9-11,18,21,24,26,29-30H,3,8,12-17H2,1-2,4-5H3/t21-,24-,26+,27+,28-/m0/s1
SMILES C=C1CC[C@]2(C)[C@@H](C)CC[C@@H](O)[C@]2(CCC=C(C)C)[C@H]1CC1=CNC2=CC=CC=C12
ORIGINAL ISOLATION REFERENCE
CITATION Gloer, James B.; Rinderknecht, Brad L.; Wicklow, Donald T.; Dowd, Patrick F. Nominine: A New Insecticidal Indole Diterpene from the Sclerotia of Aspergillus nomius Journal of Organic Chemistry 1989 54 (11) 2530-2532.
DOI 10.1021/jo00272a012 PMID -
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Eurotiomycetes MycoBank 147545
Order Eurotiales MycoBank 5042
Family Aspergillaceae MycoBank 1131492
Genus Aspergillus MycoBank 5052
SYNTHESES
CITATION 1 Peese KM; Gin DY Efficient synthetic access to the hetisine C20-diterpenoid alkaloids. A concise synthesis of nominine via oxidoisoquinolinium-1,3-dipolar and dienamine-Diels-Alder cycloadditions. Journal of the American Chemical Society 2006 128 (27) 8734-8735. DOI: 10.1021/ja0625430 PMID: 16819859
CITATION 2 Muratake H; Natsume M Total synthesis of (+/-)-nominine, a heptacyclic hetisine-type aconite alkaloid. Angewandte Chemie International Edition 2004 43 (35) 4646-4649. DOI: 10.1002/anie.200460332 PMID: 15352194
CITATION 3 Peese KM; Gin DY Asymmetric synthetic access to the hetisine alkaloids: total synthesis of (+)-nominine. Chemistry - A European Journal 2008 14 (5) 1654-1665. DOI: 10.1002/chem.200701290 PMID: 18046691
REVISIONS
VERSION SMILES CITATION
Original Isolation C[C@@H]1CC[C@@H]([C@@]2([C@]1(CCC(=C)[C@H]2CC3=CNC4=CC=CC=C43)C)CCC=C(C)C)O Gloer, James B.; Rinderknecht, Brad L.; Wicklow, Donald T.; Dowd, Patrick F. Nominine: A New Insecticidal Indole Diterpene from the Sclerotia of Aspergillus nomius Journal of Organic Chemistry 1989 54 (11) 2530-2532. DOI: 10.1021/jo00272a012
2 C=C1CC[C@]2(C)[C@@H](C)CC[C@@H](O)[C@]2(CCC=C(C)C)[C@H]1CC1=CNC2=CC=CC=C12 Bradshaw, Ben; Etxebarria-Jardí, Gorka; Bonjoch, Josep Total synthesis of (-)-anominine. Journal of the American Chemical Society 2010 132 (17) 5966-7. DOI: 10.1021/ja101994q PMID: 20384301
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