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Compounds

COMPOUND NPA018268

STRUCTURE
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PROPERTIES
NPAID NPA018268
CLUSTER ID 2157
NODE ID 1720
NAME Esperamicin A1b
FORMULA C58H78N4O22S4
MOLECULAR WEIGHT (Da) 1311.5360
ACCURATE MASS (Da) 1310.3991
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Actinomadura
ORIGIN SPECIES verrucosospora, strain H964-62
InChIKey XRUOAZDGFKHLOS-SWIZYSBBSA-N
InChI InChI=1S/C58H78N4O22S4/c1-13-59-35-27-76-42(26-39(35)72-7)81-51-48(65)46(62-84-44-25-37(64)52(85-11)30(4)78-44)28(2)79-56(51)80-38-18-16-14-15-17-20-58(70)33(19-21-87-88-86-12)45(38)47(61-57(69)75-10)49(66)53(58)82-43-24-36(63)50(29(3)77-43)83-55(68)32-22-40(73-8)41(74-9)23-34(32)60-54(67)31(5)71-6/h14-15,19,22-23,28-30,35-39,42-44,46,48,50-53,56,59,62-65,70H,5,13,21,24-27H2,1-4,6-12H3,(H,60,67)(H,61,69)/b15-14-,33-19+/t28?,29?,30?,35?,36?,37?,38-,39?,42?,43?,44?,46?,48?,50?,51?,52?,53?,56?,58+/m0/s1
SMILES CCNC1COC(CC1OC)OC2C(C(C(OC2O[C@H]3C#C/C=C\C#C[C@@]\4(C(C(=O)C(=C3/C4=C\CSSSC)NC(=O)OC)OC5CC(C(C(O5)C)OC(=O)C6=CC(=C(C=C6NC(=O)C(=C)OC)OC)OC)O)O)C)NOC7CC(C(C(O7)C)SC)O)O
ORIGINAL ISOLATION REFERENCE
CITATION KONISHI, MASATAKA; OHKUMA, HIROAKI; SAITOH, KYO-ICHIRO; KAWAGUCHI, HIROSHI; GOLIK, JERZY; DUBAY, GEORGE; GROENEWOLD, GARY; KRISHNAN, BALA; DOYLE, TERRENCE W Esperamicins, a novel class of potent antitumor antibiotics Journal of Antibiotics 1985 38 (11) 1605-1609.
DOI 10.7164/antibiotics.38.1605 PMID 4077737
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Actinobacteria LPSN 201174
Class Actinobacteria LPSN -
Order Streptosporangiales LPSN 85012
Family Thermomonosporaceae LPSN 2012
Genus Actinomadura LPSN 1988
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