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Compounds

COMPOUND NPA017432

STRUCTURE
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PROPERTIES
NPAID NPA017432
CLUSTER ID 2157
NODE ID 1720
NAME Esperamicin A1
FORMULA C59H80N4O22S4
MOLECULAR WEIGHT (Da) 1325.5630
ACCURATE MASS (Da) 1324.4147
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Actinomadura
ORIGIN SPECIES verrucosospora, strain H964-62
InChIKey LJQQFQHBKUKHIS-IIZLOWFNSA-N
InChI InChI=1S/C59H80N4O22S4/c1-28(2)60-36-27-77-43(25-39(36)73-8)83-52-50(66)47(63-85-45-24-37(64)53(86-12)31(5)79-45)29(3)80-57(52)82-38-18-16-14-15-17-20-59(71)34(19-21-88-89-87-13)46(38)48(62-58(70)76-11)51(67)54(59)84-44-26-42(49(65)30(4)78-44)81-56(69)33-22-40(74-9)41(75-10)23-35(33)61-55(68)32(6)72-7/h14-15,19,22-23,28-31,36-39,42-45,47,49-50,52-54,57,60,63-66,71H,6,21,24-27H2,1-5,7-13H3,(H,61,68)(H,62,70)/b15-14-,34-19+/t29-,30+,31-,36+,37+,38+,39+,42+,43+,44+,45+,47-,49-,50+,52-,53-,54-,57+,59-/m1/s1
SMILES C=C(OC)C(=O)NC1=CC(OC)=C(OC)C=C1C(=O)O[C@H]1C[C@H](O[C@@H]2C(=O)C(NC(=O)OC)=C3/C(=C\CSSSC)[C@]2(O)C#C/C=C\C#C[C@@H]3O[C@@H]2O[C@H](C)[C@@H](NO[C@H]3C[C@H](O)[C@H](SC)[C@@H](C)O3)[C@H](O)[C@H]2O[C@H]2C[C@H](OC)[C@@H](NC(C)C)CO2)O[C@@H](C)[C@H]1O
ORIGINAL ISOLATION REFERENCE
CITATION KONISHI, MASATAKA; OHKUMA, HIROAKI; SAITOH, KYO-ICHIRO; KAWAGUCHI, HIROSHI; GOLIK, JERZY; DUBAY, GEORGE; GROENEWOLD, GARY; KRISHNAN, BALA; DOYLE, TERRENCE W Esperamicins, a novel class of potent antitumor antibiotics Journal of Antibiotics 1985 38 (11) 1605-1609.
DOI 10.7164/antibiotics.38.1605 PMID 4077737
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Actinobacteria LPSN 201174
Class Actinobacteria LPSN -
Order Streptosporangiales LPSN 85012
Family Thermomonosporaceae LPSN 2012
Genus Actinomadura LPSN 1988
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