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Compounds

COMPOUND NPA016780

STRUCTURE
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PROPERTIES
NPAID NPA016780
CLUSTER ID 5702
NODE ID 4035
NAME Balanol
FORMULA C28H26N2O10
MOLECULAR WEIGHT (Da) 550.5200
ACCURATE MASS (Da) 550.1587
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Verticillium
ORIGIN SPECIES balanoides
InChIKey XYUFCXJZFZPEJD-XMSQKQJNSA-N
InChI InChI=1S/C28H26N2O10/c31-16-8-6-14(7-9-16)26(36)30-18-13-29-10-2-5-22(18)40-28(39)15-11-20(33)24(21(34)12-15)25(35)23-17(27(37)38)3-1-4-19(23)32/h1,3-4,6-9,11-12,18,22,29,31-34H,2,5,10,13H2,(H,30,36)(H,37,38)/t18-,22-/m1/s1
SMILES C1C[C@H]([C@@H](CNC1)NC(=O)C2=CC=C(C=C2)O)OC(=O)C3=CC(=C(C(=C3)O)C(=O)C4=C(C=CC=C4O)C(=O)O)O
ORIGINAL ISOLATION REFERENCE
CITATION Kulanthaivel, Palaniappan; Hallock, Yali F.; Boros, Christie; Hamilton, Sean M.; Janzen, William P.; Ballas, Lawrence M.; Loomis, Carson R.; Jiang, Jack B.; Katz, Barry Balanol: a novel and potent inhibitor of protein kinase C from the fungus Verticillium balanoides Journal of the American Chemical Society 1993 115 (14) 6452-6453.
DOI 10.1021/ja00067a087 PMID -
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Sordariomycetes MycoBank 147550
Order Glomerellales MycoBank 1028384
Family Plectosphaerellaceae MycoBank 1033978
Genus Verticillium MycoBank 1036719
SYNTHESES
CITATION 1 Fürstner A; Thiel OR Formal total synthesis of (-)-balanol: concise approach to the hexahydroazepine segment based on RCM. Journal of Organic Chemistry 2000 65 (6) 1738-42. DOI: 10.1021/jo991611g PMID: 10750493
CITATION 2 Lampe JW; Hughes PF; Biggers CK; Smith SH; Hu H Total Synthesis of (-)- and (+)-Balanol(1). Journal of Organic Chemistry 1996 61 (14) 4572-4581. DOI: 10.1021/jo952280k PMID: 11667382
CITATION 3 Srivastava AK; Panda G Total synthesis of (-)-balanol, all stereoisomers, their N-tosyl analogues, and fully protected ophiocordin: an easy route to hexahydroazepine cores from garner aldehydes. Chemistry - A European Journal 2008 14 (15) 4675-88. DOI: 10.1002/chem.200701991 PMID: 18399526
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