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Compounds

COMPOUND NPA015291

STRUCTURE
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EXTERNAL LINKS
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PROPERTIES
NPAID NPA015291
CLUSTER ID 3188
NODE ID 2427
NAME Urukthapelstatin A
FORMULA C34H30N8O6S2
MOLECULAR WEIGHT (Da) 710.7980
ACCURATE MASS (Da) 710.1730
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Mechercharimyces
ORIGIN SPECIES asporophorigenens YM11-542
InChIKey LDFMSIKUSPHBGH-GTAKYJCGSA-N
InChI InChI=1S/C34H30N8O6S2/c1-5-16(3)24-28(44)35-17(4)27(43)36-19(6-2)30-37-20(12-46-30)31-38-21(13-47-31)33-40-23(15-50-33)34-39-22(14-49-34)32-42-25(29(45)41-24)26(48-32)18-10-8-7-9-11-18/h6-17,24H,5H2,1-4H3,(H,35,44)(H,36,43)(H,41,45)/b19-6-/t16-,17-,24+/m0/s1
SMILES CC[C@H](C)[C@@H]1C(=O)N[C@H](C(=O)N/C(=C\C)/C2=NC(=CO2)C3=NC(=CO3)C4=NC(=CS4)C5=NC(=CS5)C6=NC(=C(O6)C7=CC=CC=C7)C(=O)N1)C
ORIGINAL ISOLATION REFERENCE
CITATION Matsuo, Yoshihide; Kanoh, Kaneo; Imagawa, Hiroshi; Adachi, Kyoko; Nishizawa, Mugio; Shizuri, Yoshikazu Urukthapelstatin A, a Novel Cytotoxic Substance from Marine-derived Mechercharimyces asporophorigenens YM11-542 Journal of Antibiotics 2007 60 (4) 256-260.
DOI 10.1038/ja.2007.31 PMID 17456976
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Firmicutes LPSN 1239
Class Bacilli LPSN 91061
Order Bacillales LPSN 1385
Family Thermoactinomycetaceae LPSN 186824
Genus Mechercharimyces LPSN 482144
SYNTHESES
CITATION 1 Lin CC; Tantisantisom W; McAlpine SR Total synthesis and biological activity of natural product Urukthapelstatin A. Organic Letters 2013 15 (14) 3574-7. DOI: 10.1021/ol401412v PMID: 23819711
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