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Compounds

COMPOUND NPA012028

STRUCTURE
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EXTERNAL LINKS
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PROPERTIES
NPAID NPA012028
CLUSTER ID 26
NODE ID 25
NAME Apicidin C
FORMULA C33H47N5O6
MOLECULAR WEIGHT (Da) 609.7680
ACCURATE MASS (Da) 609.3526
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Fusarium
ORIGIN SPECIES sp.
InChIKey GWLHFNKLJRZBAI-KGKLHAENSA-N
InChI InChI=1S/C33H47N5O6/c1-5-23(39)13-7-6-8-15-25-30(40)35-26(19-22-20-38(44-4)27-16-10-9-14-24(22)27)31(41)36-29(21(2)3)33(43)37-18-12-11-17-28(37)32(42)34-25/h9-10,14,16,20-21,25-26,28-29H,5-8,11-13,15,17-19H2,1-4H3,(H,34,42)(H,35,40)(H,36,41)/t25-,26-,28+,29-/m0/s1
SMILES CCC(=O)CCCCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N2CCCC[C@@H]2C(=O)N1)C(C)C)CC3=CN(C4=CC=CC=C43)OC
ORIGINAL ISOLATION REFERENCE
CITATION Singh, Sheo B.; Zink, Deborah L.; Liesch, Jerrold M.; Mosley, Ralph T.; Dombrowski, Anne W.; Bills, Gerald F.; Darkin-Rattray, Sandra J.; Schmatz, Dennis M.; Goetz, Michael A. Structure and chemistry of apicidins, a class of novel cyclic tetrapeptides without a terminal α-keto epoxide as inhibitors of histone deacetylase with potent antiprotozoal activities Journal of Organic Chemistry 2002 67 (3) 815-825.
DOI 10.1021/jo016088w PMID 11856024
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Sordariomycetes MycoBank 147550
Order Hypocreales MycoBank 5125
Family Nectriaceae MycoBank 110618
Genus Fusarium MycoBank 5506
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