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Compounds

COMPOUND NPA011301

STRUCTURE
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PROPERTIES
NPAID NPA011301
CLUSTER ID 3833
NODE ID 2872
NAME Calphostin D
FORMULA C30H30O10
MOLECULAR WEIGHT (Da) 550.5600
ACCURATE MASS (Da) 550.1839
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Cladosporium
ORIGIN SPECIES cladosporioides
InChIKey WJBHEYCJMSCKIP-UHFFFAOYSA-N
InChI InChI=1S/C30H30O10/c1-11(31)7-13-19-20-14(8-12(2)32)30(40-6)28(36)22-16(34)10-18(38-4)24(26(20)22)23-17(37-3)9-15(33)21(25(19)23)27(35)29(13)39-5/h9-12,31-32,35-36H,7-8H2,1-6H3
SMILES CC(CC1=C(C(=C2C(=O)C=C(C3=C4C(=CC(=O)C5=C(C(=C(C(=C45)C1=C32)CC(C)O)OC)O)OC)OC)O)OC)O
ORIGINAL ISOLATION REFERENCE
CITATION Kobayashi; Ando; Nakano; Iida; Ohno; Morimoto; Tamaoki Calphostins (UCN-1028), novel and specific inhibitors of protein kinase C. I. Fermentation, isolation, physico-chemical properties and biological activities Journal of Antibiotics 1989 42 (10) 1470-1474.
DOI 10.7164/antibiotics.42.1470 PMID 2478514
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Dothideomycetes MycoBank 147541
Order Capnodiales MycoBank 134362
Family Cladosporiaceae MycoBank 452563
Genus Cladosporium MycoBank 5498
SYNTHESES
CITATION 1 Morgan BJ; Mulrooney CA; O'Brien EM; Kozlowski MC Perylenequinone natural products: total syntheses of the diastereomers (+)-phleichrome and (+)-calphostin D by assembly of centrochiral and axial chiral fragments. Journal of Organic Chemistry 2010 75 (1) 30-43. DOI: 10.1021/jo901384h PMID: 19894745
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