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Compounds

COMPOUND NPA011020

STRUCTURE
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PROPERTIES
NPAID NPA011020
CLUSTER ID 283
NODE ID 257
NAME Microcin SF608
FORMULA C32H44N6O6
MOLECULAR WEIGHT (Da) 608.7400
ACCURATE MASS (Da) 608.3322
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Microcystis
ORIGIN SPECIES sp.
InChIKey HYPWKJJQJSEUDS-GFZBRZDVSA-N
InChI InChI=1S/C32H44N6O6/c33-32(34)36-15-5-4-14-35-29(42)27-18-22-10-13-24(40)19-26(22)38(27)31(44)25(16-20-6-2-1-3-7-20)37-30(43)28(41)17-21-8-11-23(39)12-9-21/h1-3,6-9,11-12,22,24-28,39-41H,4-5,10,13-19H2,(H,35,42)(H,37,43)(H4,33,34,36)/t22-,24+,25-,26-,27-,28-/m0/s1
SMILES C1C[C@H](C[C@H]2[C@@H]1C[C@H](N2C(=O)[C@H](CC3=CC=CC=C3)NC(=O)[C@H](CC4=CC=C(C=C4)O)O)C(=O)NCCCCN=C(N)N)O
ORIGINAL ISOLATION REFERENCE
CITATION Banker, Ronny; Carmeli, Shmuel Inhibitors of serine proteases from a waterbloom of the cyanobacterium Microcystis sp Tetrahedron 1999 55 (35) 10835-10844.
DOI 10.1016/s0040-4020(99)00597-9 PMID -
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Cyanobacteria LPSN 1117
Class Cyanophyceae LPSN -
Order Chroococcales LPSN 1118
Family Microcystaceae LPSN 1890449
Genus Microcystis LPSN 1125
SYNTHESES
CITATION 1 Diethelm S; Schindler CS; Carreira EM Access to the aeruginosin serine protease inhibitors through the nucleophilic opening of an oxabicyclo[2.2.1]heptane: total synthesis of microcin SF608. Chemistry - A European Journal 2014 20 (20) 6071-6080. DOI: 10.1002/chem.201400046 PMID: 24687726
CITATION 2 Diethelm S; Schindler CS; Carreira EM Synthesis of Microcin SF608 through nucleophilic opening of an oxabicyclo[2.2.1]heptane. Organic Letters 2010 12 (17) 3950-3953. DOI: 10.1021/ol1017189 PMID: 20704315
CITATION 3 Valls N; Vallribera M; López-Canet M; Bonjoch J Synthesis of microcin SF608. Journal of Organic Chemistry 2002 67 (14) 4945-4950. DOI: 10.1021/jo025709y PMID: 12098309
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