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Compounds

COMPOUND NPA010319

STRUCTURE
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PROPERTIES
NPAID NPA010319
CLUSTER ID 739
NODE ID 645
NAME Spliceostatin G
FORMULA C21H31NO6
MOLECULAR WEIGHT (Da) 393.4800
ACCURATE MASS (Da) 393.2151
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Burkholderia
ORIGIN SPECIES sp. FERM BP-3421
InChIKey SPJBXWLUCQGFSA-OGGYWXJKSA-N
InChI InChI=1S/C21H31NO6/c1-13(7-11-21(25)26)6-9-19-14(2)12-18(16(4)28-19)22-20(24)10-8-15(3)27-17(5)23/h6-8,10-11,14-16,18-19H,9,12H2,1-5H3,(H,22,24)(H,25,26)/b10-8-,11-7+,13-6+/t14-,15-,16+,18+,19-/m0/s1
SMILES C[C@H]1C[C@H]([C@H](O[C@H]1C/C=C(\C)/C=C/C(=O)O)C)NC(=O)/C=C\[C@H](C)OC(=O)C
ORIGINAL ISOLATION REFERENCE
CITATION He, Haiyin; Ratnayake, Anokha S.; Janso, Jeffrey E.; He, Min; Yang, Hui Y.; Loganzo, Frank; Shor, Boris; O'Donnell, Christopher J.; Koehn, Frank E. Cytotoxic spliceostatins from Burkholderia sp. and their semisynthetic analogues Journal of Natural Products 2014 77 (8) 1864-1870.
DOI 10.1021/np500342m PMID 25098528
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Proteobacteria LPSN 1224
Class Betaproteobacteria LPSN 28216
Order Burkholderiales LPSN 80840
Family Burkholderiaceae LPSN 119060
Genus Burkholderia LPSN 32008
SYNTHESES
CITATION 1 Ghosh AK; Reddy GC; MacRae AJ; Jurica MS Enantioselective Synthesis of Spliceostatin G and Evaluation of Bioactivity of Spliceostatin G and Its Methyl Ester. Organic Letters 2018 20 (1) 96-99. DOI: 10.1021/acs.orglett.7b03456 PMID: 29218995
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