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Compounds

COMPOUND NPA008028

STRUCTURE
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PROPERTIES
NPAID NPA008028
CLUSTER ID 22
NODE ID 21
NAME Aigialomycin D
FORMULA C18H22O6
MOLECULAR WEIGHT (Da) 334.3680
ACCURATE MASS (Da) 334.1416
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Aigialus
ORIGIN SPECIES parvus BCC 5311
InChIKey NHAQNKDEUQPSIX-DXOCLGOBSA-N
InChI InChI=1S/C18H22O6/c1-11-5-4-8-15(21)14(20)7-3-2-6-12-9-13(19)10-16(22)17(12)18(23)24-11/h2,4,6,8-11,14-15,19-22H,3,5,7H2,1H3/b6-2+,8-4+/t11-,14-,15+/m0/s1
SMILES C[C@H]1C/C=C/[C@H]([C@H](CC/C=C/C2=CC(=CC(=C2C(=O)O1)O)O)O)O
ORIGINAL ISOLATION REFERENCE
CITATION Isaka, Masahiko; Suyarnsestakorn, Chotika; Tanticharoen, Morakot; Kongsaeree, Palangpon; Thebtaranonth, Yodhathai Aigialomycins A-E, new resorcylic macrolides from the marine mangrove fungus Aigialus parvus Journal of Organic Chemistry 2002 67 (5) 1561-1566.
DOI 10.1021/jo010930g PMID 11871887
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Dothideomycetes MycoBank 147541
Order Pleosporales MycoBank 92860
Family Aigialaceae MycoBank 715274
Genus Aigialus MycoBank 193126
SYNTHESES
CITATION 1 Calo F; Richardson J; Barrett AG Total synthesis of aigialomycin D using a one-pot ketene generation-trapping-aromatization sequence. Organic Letters 2009 11 (21) 4910-4913. DOI: 10.1021/ol901979x PMID: 19799447
CITATION 2 Chrovian CC; Knapp-Reed B; Montgomery J Total synthesis of aigialomycin D: surprising chemoselectivity dependence on alkyne structure in nickel-catalyzed cyclizations. Organic Letters 2008 10 (5) 811-814. DOI: 10.1021/ol702961v PMID: 18254635
CITATION 3 Baird LJ; Timmer MS; Teesdale-Spittle PH; Harvey JE Total synthesis of aigialomycin D using a Ramberg-Bäcklund/RCM strategy. Journal of Organic Chemistry 2009 74 (6) 2271-2277. DOI: 10.1021/jo802561s PMID: 19284735
CITATION 4 Geng X; Danishefsky SJ Total synthesis of aigialomycin D. Organic Letters 2004 6 (3) 413-416. DOI: 10.1021/ol036258m PMID: 14748606
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