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Compounds

COMPOUND NPA004614

STRUCTURE
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PROPERTIES
NPAID NPA004614
CLUSTER ID 249
NODE ID 228
NAME Sphingofungin F
FORMULA C21H39NO6
MOLECULAR WEIGHT (Da) 401.5440
ACCURATE MASS (Da) 401.2777
ORIGIN ORGANISM TYPE Fungus
ORIGIN GENUS Paecilomyces
ORIGIN SPECIES variotii
InChIKey KEACSJIKRANUJC-NZBAJYJFSA-N
InChI InChI=1S/C21H39NO6/c1-3-4-5-10-13-16(23)14-11-8-6-7-9-12-15-17(24)18(25)19(26)21(2,22)20(27)28/h12,15,17-19,24-26H,3-11,13-14,22H2,1-2H3,(H,27,28)/b15-12+/t17-,18+,19-,21-/m0/s1
SMILES CCCCCCC(=O)CCCCCC/C=C/[C@H](O)[C@@H](O)[C@H](O)[C@](C)(N)C(=O)O
ORIGINAL ISOLATION REFERENCE
CITATION Horn, W S; Smith, J L; Bills, G F; Raghoobar, S L; Helms, G L; Kurtz, M B; Marrinan, J A; Frommer, B R; Thornton, R A; Mandala, S M Sphingofungins E and F: novel serinepalmitoyl transferase inhibitors from Paecilomyces variotii. Journal of Antibiotics 1992 45 (10) 1692-1696.
DOI 10.7164/antibiotics.45.1692 PMID 1474000
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Eukarya - 2759
Kingdom Fungi MycoBank 4751
Phylum Ascomycota MycoBank 4890
Class Eurotiomycetes MycoBank 147545
Order Eurotiales MycoBank 5042
Family Trichocomaceae MycoBank 28568
Genus Paecilomyces MycoBank 33202
SYNTHESES
CITATION 1 Lee KY; Oh CY; Ham WH Total synthesis of sphingofungin F. Organic Letters 2002 4 (25) 4403-5. DOI: 10.1021/ol020164f PMID: 12465898
CITATION 2 Gan FF; Yang SB; Luo YC; Yang WB; Xu PF Total synthesis of sphingofungin F based on chiral tricyclic iminolactone. Journal of Organic Chemistry 2010 75 (8) 2737-40. DOI: 10.1021/jo100183d PMID: 20329736
CITATION 3 Tsuzaki S; Usui S; Oishi H; Yasushima D; Fukuyasu T; Oishi T; Sato T; Chida N Total synthesis of sphingofungin F by orthoamide-type overman rearrangement of an unsaturated ester. Organic Letters 2015 17 (7) 1704-7. DOI: 10.1021/acs.orglett.5b00475 PMID: 25769012
REVISIONS
VERSION SMILES CITATION
Original Isolation CCCCCCC(=O)CCCCCC/C=C/C(C(C(C(C)(C(=O)O)N)O)O)O Horn, W S; Smith, J L; Bills, G F; Raghoobar, S L; Helms, G L; Kurtz, M B; Marrinan, J A; Frommer, B R; Thornton, R A; Mandala, S M Sphingofungins E and F: novel serinepalmitoyl transferase inhibitors from Paecilomyces variotii. Journal of Antibiotics 1992 45 (10) 1692-1696. DOI: 10.7164/antibiotics.45.1692 PMID: 1474000
2 CCCCCCC(=O)CCCCCC/C=C/[C@H](O)[C@@H](O)[C@H](O)[C@](C)(N)C(=O)O Tsuzaki S; Usui S; Oishi H; Yasushima D; Fukuyasu T; Oishi T; Sato T; Chida N Total synthesis of sphingofungin F by orthoamide-type overman rearrangement of an unsaturated ester. Organic Letters 2015 17 (7) 1704-7. DOI: 10.1021/acs.orglett.5b00475 PMID: 25769012
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