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Compounds

COMPOUND NPA003100

STRUCTURE
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PROPERTIES
NPAID NPA003100
CLUSTER ID 1762
NODE ID 1429
NAME Cycloviracin B1
FORMULA C83H152O33
MOLECULAR WEIGHT (Da) 1678.0960
ACCURATE MASS (Da) 1677.0216
ORIGIN ORGANISM TYPE Bacterium
ORIGIN GENUS Kibdelosporangium
ORIGIN SPECIES albatum No. R 761-7
InChIKey UHXMKKIXCMBBAY-NFPDUFFVSA-N
InChI InChI=1S/C83H152O33/c1-51(87)36-28-26-34-40-53(108-82-77(103-4)72(98)65(91)58(47-85)113-82)38-30-22-19-15-12-9-13-17-21-25-33-43-56-45-63(89)106-50-60-67(93)69(95)74(100)79(115-60)110-55(44-62(88)105-49-61-68(94)70(96)75(101)80(111-56)116-61)42-32-24-20-16-11-8-6-7-10-14-18-23-31-39-54(109-83-78(104-5)73(99)66(92)59(48-86)114-83)41-35-27-29-37-52(2)107-81-76(102-3)71(97)64(90)57(46-84)112-81/h51-61,64-87,90-101H,6-50H2,1-5H3/t51?,52?,53?,54?,55-,56-,57?,58?,59?,60?,61?,64?,65?,66?,67?,68?,69?,70?,71?,72?,73?,74?,75?,76?,77?,78?,79?,80?,81?,82?,83?/m1/s1
SMILES COC1C(OC(C)CCCCCC(CCCCCCCCCCCCCCC[C@@H]2CC(=O)OCC3OC(O[C@H](CCCCCCCCCCCCCC(CCCCCC(C)O)OC4OC(CO)C(O)C(O)C4OC)CC(=O)OCC4OC(O2)C(O)C(O)C4O)C(O)C(O)C3O)OC2OC(CO)C(O)C(O)C2OC)OC(CO)C(O)C1O
ORIGINAL ISOLATION REFERENCE
CITATION TSUNAKAWA, MITSUAKI; KOTAKE, CHIKAKO; YAMASAKI, TETSURO; MORIYAMA, TOSHIO; KONISHI, MASATAKA; OKI, TOSHIKAZU New antiviral antibiotics, cycloviracins B1 and B2. II. Structure determination Journal of Antibiotics 1992 45 (9) 1472-1480.
DOI 10.7164/antibiotics.45.1472 PMID 1429233
ORIGINAL ISOLATION TAXONOMY
RANK NAME DB LINK NCBI
Domain Bacteria LPSN 2
Phylum Actinobacteria LPSN 201174
Class Actinobacteria LPSN -
Order Pseudonocardiales LPSN 85010
Family Pseudonocardiaceae LPSN 2070
Genus Kibdelosporangium LPSN 2029
SYNTHESES
CITATION 1 Fürstner A; Albert M; Mlynarski J; Matheu M; DeClercq E Structure assignment, total synthesis, and antiviral evaluation of cycloviracin B1. Journal of the American Chemical Society 2003 125 (43) 13132-42. DOI: 10.1021/ja036521e PMID: 14570487
REVISIONS
VERSION SMILES CITATION
Original Isolation CC(CCCCCC(CCCCCCCCCCCCCC1CC(=O)OCC2C(C(C(C(O2)OC(CC(=O)OCC3C(C(C(C(O1)O3)O)O)O)CCCCCCCCCCCCCCCC(CCCCCC(C)OC4C(C(C(C(O4)CO)O)O)OC)OC5C(C(C(C(O5)CO)O)O)OC)O)O)O)OC6C(C(C(C(O6)CO)O)O)OC)O TSUNAKAWA, MITSUAKI; KOTAKE, CHIKAKO; YAMASAKI, TETSURO; MORIYAMA, TOSHIO; KONISHI, MASATAKA; OKI, TOSHIKAZU New antiviral antibiotics, cycloviracins B1 and B2. II. Structure determination Journal of Antibiotics 1992 45 (9) 1472-1480. DOI: 10.7164/antibiotics.45.1472 PMID: 1429233
2 COC1C(OC(C)CCCCCC(CCCCCCCCCCCCCCC[C@@H]2CC(=O)OCC3OC(O[C@H](CCCCCCCCCCCCCC(CCCCCC(C)O)OC4OC(CO)C(O)C(O)C4OC)CC(=O)OCC4OC(O2)C(O)C(O)C4O)C(O)C(O)C3O)OC2OC(CO)C(O)C(O)C2OC)OC(CO)C(O)C1O Fürstner, Alois; Albert, Martin; Mlynarski, Jacek; Matheu, Maribel A concise synthesis of the fully functional lactide core of cycloviracin B with implications for the structural assignment of related glycolipids. Journal of the American Chemical Society 2002 124 (7) 1168-9. DOI: 10.1021/ja0175791 PMID: 11841275
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